Question:medium

Which oral hypoglycemic agent increases the levels of incretin hormone by inhibiting the enzyme dipeptidyl peptidase-4 (DPP-4):

Show Hint

Sitagliptin is a DPP-4 inhibitor that boosts incretin levels, enhancing insulin secretion and improving glucose control in patients with type 2 diabetes.
Updated On: Jul 14, 2026
  • Metformin
  • Pioglitazone
  • Sitagliptin
  • Glipizide
Show Solution

The Correct Option is C

Solution and Explanation

Step 1: Understanding the Question:
We need to pick the oral anti-diabetic drug that works by blocking DPP-4, an enzyme that breaks down incretin hormones.

Step 2: Key Concept:
Drugs ending in "-gliptin" belong to the DPP-4 inhibitor class. DPP-4 normally degrades GLP-1 and GIP within minutes; stopping this enzyme keeps incretin levels high, which increases insulin release after meals.

Step 3: Detailed Explanation:
Metformin is a biguanide that reduces liver glucose output. Pioglitazone is a thiazolidinedione that improves insulin sensitivity through PPAR-gamma activation. Glipizide is a sulfonylurea that forces insulin release by blocking potassium channels on beta cells. None of these three touch DPP-4. Sitagliptin, by contrast, is named with the "-gliptin" suffix and is a direct DPP-4 inhibitor, matching the mechanism described in the question exactly.

Step 4: Final Answer:
The drug that raises incretin levels by inhibiting DPP-4 is Sitagliptin.
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