Question:medium

Which of the following is peroxisome proliferator-activated receptor-alpha (PPAR-α) agonist:

Updated On: Jul 14, 2026
  • Ezetimibe
  • Niacin
  • Colesevelam
  • Gemfibrozil
Show Solution

The Correct Option is D

Solution and Explanation

Each of the four drugs listed belongs to a distinct class of lipid-lowering agent with its own separate mechanism: ezetimibe blocks cholesterol absorption at the intestinal brush border, niacin acts through an adipose-tissue receptor to reduce fat breakdown, and colesevelam binds and removes bile acids to indirectly lower cholesterol. Fibrates, the class gemfibrozil belongs to, are the one group of lipid-lowering drugs whose mechanism is built specifically around activating the PPAR-α nuclear receptor in liver and muscle tissue, which switches on genes for fatty acid oxidation and lipoprotein lipase, ultimately lowering triglycerides.

Therefore, the correct answer is Gemfibrozil.

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